The present invention provides cancer treatment preparations of excellent targetability. The sugar chain-modified liposomes of the present invention,which contain an aromatase inhibitor,anti-androgenic agent, lyase inhibitor,GnRH agonist,GnRH antagonist,anti-angiogenic agent,tyrosine kinase inhibitor,serine-threonine kinase inhibitor,antibody having an anticancer activity,ansamitocin,capecitabine, celmoleukin,docetaxel hydrate, gemcitabine hydrochloride,oxaliplatin,prednisolone,tegafur-uracil mixtures,zinostatin stimalamer or arsenic trioxide may be used as cancer treatment preparations having an excellent targetability.